Title | ||
---|---|---|
2-Furoic piperazide derivatives as promising drug candidates of type 2 diabetes and Alzheimer's diseases: In vitro and in silico studies. |
Abstract | ||
---|---|---|
•Synthesis of multi-functional 2-furoic piperazide derivatives.•Enzyme inhibitory studies against different enzymes.•Computational studies to augment the in vitro results.•Suitable therapeutic agents for type 2 diabetes and Alzheimer’s disease.•Mild hemolytic agents toward red blood cell membrane. |
Year | DOI | Venue |
---|---|---|
2018 | 10.1016/j.compbiolchem.2018.09.007 | Computational Biology and Chemistry |
Keywords | Field | DocType |
2-Furoic piperazide,Sulfonamide,Enzyme inhibition,Molecular docking,α-Glucosidase,Cholinesterases | Acetylcholinesterase,Docking (molecular),Drug discovery,Enzyme,Biology,In vitro,Combinatorial chemistry,Acarbose,Butyrylcholinesterase,Genetics,Piperazine | Journal |
Volume | ISSN | Citations |
77 | 1476-9271 | 0 |
PageRank | References | Authors |
0.34 | 4 | 9 |
Name | Order | Citations | PageRank |
---|---|---|---|
Muhammad Athar Abbasi | 1 | 0 | 0.34 |
Mubashir Hassan | 2 | 0 | 0.68 |
Aziz ur-Rehman | 3 | 0 | 0.34 |
Sabahat Zahra Siddiqui | 4 | 0 | 0.34 |
Ghulam Hussain | 5 | 0 | 0.34 |
Syed Adnan Ali Shah | 6 | 0 | 0.34 |
Muhammad Ashraf | 7 | 7 | 4.62 |
Muhammad Shahid | 8 | 25 | 8.75 |
Y. Sung | 9 | 13 | 1.85 |